 Antiallergic agent |
| What is claimed is: 1. A method for the treatment and prevention of allergic diseases, comprising ... |
|
| Hyaluronate-poly (ethylene oxide) compositions and cosmetic formulations thereof |
| OF THE INVENTION As noted above, the invention provides highly viscoelastic compositions ... |
|
| Antiviral compounds |
| We claim: 1. A compound of formula (I)B ##STR7## wherein R.sup.1 represents an oxo or imino group; R... |
|
| Process for the production of 2-equivalent yellow couplers |
| I claim: 1. In the process of converting a photographic 4-equivalent acyl acetamide yellow coupler ... |
|
| Triazinyl-antraquinone dyes |
| What is claimed is: 1. A compound of the formula ##STR63## wherein R and R' each are hydrogen, C.... |
|
| 6-Fluoro-3,5-dichloro-2-pyridinyl phosphorus compounds |
| What is claimed is: 1. A compound corresponding to the formula ##STR6## wherein R represents alkyl ... |
|
| Stabilized insecticide formulations |
| What is claimed is: 1. In a solid stabilized insecticidal composition mixture which comprises from ... |
|
|
Cyclopropane carboxylic acid derivatives
| Details |
|
Inventors: Tessier, Jean; Demoute, Jean-Pierre; Cadiergue, Joseph;
Assignee: Roussel Uclaf (Paris, FR)
Primary Examiner:
Assistant Examiner:
Attorney, Agent or Firm:
All stereoisomeric forms and mixtures of stereoisomers of compounds of the formula ##STR1## wherein X is selected from the group consisting of oxygen, sulfur, sulfoxide and sulfone, R.sub.1 and R.sub.3 are individually selected from the group consisting of optionally unsaturated alkyl of 1 to 7 carbon atoms and optionally unsaturated cycloalkyl of 3 to 7 carbon atoms optionally substituted with at least one halogen and optionally interrupted with at least one heteroatom and aryl and aralkyl of 6 to 18 carbon atoms and R.sub.2 is the residue of a R.sub.2 OH alcohol used in pyrethrinoids synthesis having pesticidal activity and their preparation and novel intermediates. |
|
DETAILED DESCRIPTION What we claim is: 1.
A compound selected from the group consisting of all stereoisomer forms and mixtures of stereoisomers of compounds of the formula ##STR25## wherein X is selected from the group consisting of oxygen, sulfur, sulfoxide and sulfone, R.
sub.
1 and R.
sub.
3 are individually selected from the group consisting of alkyl of 1 to 7 carbon atoms, alkenyl and alkadienyl of 2 to 7 carbon atoms and cycloalkyl and cycloalkenyl of 3 to 7 carbon atoms optionally substituted with at least one halogen and optionally interrupted with at least one heteroatom and aryl and aralkyl of 6 to 18 carbon atoms and R.
sub.
2 is selected from the group consisting of ##STR26## 2.
A compound of claim 1 wherein X is oxygen.
3.
A compound of claim 1 wherein X is sulfur.
4.
A compound of claim 1 selected from the group consisting of (S).
alpha.
-cyano-3-phenoxy-benzyl (1R,trans,.
DELTA.
Z) 2,2-dimethyl-3-dimethyl-3-[2-methoxy-2-methoxycarbonyl-ethenyl]-cyclopropa ne-carboxylate, (S).
alpha.
-cyano-3-phenoxy-benzyl (1R,trans,.
DELTA.
Z) 2,2-dimethyl-3-[2-methoxy-2-methoxycarbonyl-ethenyl]-cyclopropane-carboxyl ate, 3-allyl-2-methyl-4-oxo-2-cyclopenten-1-yl (1R,trans,.
DELTA.
Z) 2,2-dimethyl-3-[2-methoxy-2-methoxycarbonyl-ethenyl]-cyclopropane-carboxyl ate, 3-alkyl-2-methyl-4-oxo-2-cyclopenten-1-yl (1R, trans,.
DELTA.
E) 2,2-dimethyl-3-[2-methoxy-2-methoxycarbonyl-ethenyl]-cyclopropane-carboxyl ate, [1-(3-propyn-2-yl)-2,5-dioxo-imidazolidinyl]-methyl (1R,trans,.
DELTA.
Z) 2,2-dimethyl-3-[2-methoxy-2-methoxycarbonyl-ethenyl]-c yclopropane-carboxylate, (S).
alpha.
-cyano-3-phenoxy-4-fluoro-benzyl (1R, trans,.
DELTA.
Z or .
DELTA.
E) 2,2-dimethyl-3-[2-methoxy-2methoxycarbonyl-ethenyl]-cyclopropane-carboxyla te, (R,S).
alpha.
-cyano-6'-phenoxy-2'-pyridyl-methyl (1R,trans,.
DELTA.
Z or .
DELTA.
E) 2,2-dimethyl -3-[2-methoxy-2-methoxycarbonyl-ethenyl]-cyclopropane-carboxylate, (S).
alpha.
-cyano-3-phenoxy-benzyl (1R,trans,.
DELTA.
Z) 2,2-dimethyl-3-[2-methoxy-2-ethoxycarbonyl-ethenyl]-cyclopropane-carboxyla te, (S).
alpha.
-cyano-3-phenoxy-benzyl (1R,trans,
|
| Related patents |
|
|
Cyanovinyl pyrethroids and pesticidal use thereof
I claim: 1. A compound of the formula: ##STR151## wherein R.sub.1 is ##STR152## R.sub.3 is hydrogen or methyl; and X and X' are each hydrogen, halogen, C.sub.1 -C.sub.3 ...
|
|
|
Vaccines against feline leukemia
What is claimed is: 1. A vaccine for the prevention of disease caused by Feline leukemia virus which comprises in unit dosage form about 10.sup.7 -10.sup.9 cells ...
|
|
|
Arylethers and pharmaceutical compositions
What we claim is: 1. The aryloxy lower alkyl piperidines selected from the group consisting of -N-(2,6 dichlorophenoxy) ethyl 4-(N'-phenyl N'-propionylamino) piperidine; ...
|
|
|
1,2,4-Dihydrotriazine-4-oxides and a process for their production
We claim: 1. 1,2,4-Dihydrotriazine-4-oxides of the formula ##STR13## wherein R.sup.1 is an alkylene of 2 to 10 carbon atoms, R.sup.2 and R.sup.3 are identical or ...
|
|
|
Acid addition salts of dextrorotatory ergot alkaloids, a process for the preparation thereof as well as their use as medicines
What is claimed is: 1. A process for the treatment of a condition selected from the group of arterial hypertension, heart insufficiency, heart arrhythmia or cephalalgia, ...
|
|
|
Process for flameproofing polyurethanes
We claim: 1. An improved process for flameproofing polyurethanes using 1 to 15 percent by weight based on the polyurethane of a reactive phosphonate as flameproofing ...
|
|
|
Anabolic-weight-gain promoting compositions containing isoflavone derivatives and method using same
We claim: 1. An anabolic treatment method for human patients comprising administering to said patients in a daily dosage of 0.2 to 100 mg/kg of body weight a compound ...
|
|
|
Bridged oxygen analogs of daunorubcin and doxorubicin
We claim: 1. A compound of the formula ##STR7## wherein R is selected from the group consisting of --COCH.sub.3, --CHOHCH.sub.3, --COCH.sub.2 OH, --CHOHCH.sub.2 OH, ...
|
|
|
O-Alkyl-S-alkyl-S-branched alkylphosphorodithioate soil insecticides
What is claimed is: 1. A method for controlling corn rootworm which comprises applying to its habitat, in an amount effective for controlling corn rootworm, a compound ...
|
|
|
Process for the preparation of 2-(4-isobutylphenyl)-propiohydroxamic acid
What is claimed is: 1. A process for the preparation of 2-(4isobutylphenyl)-propiohydroxamic acid comprising the steps of forming a mixture of 2-(4-isobutylphenyl)-...
|
|
|
Vasodialators 
