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| Latest patents |
Results: 181-210 of 1119
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Method of protecting plants from pathogens with cyanomethyl aryl sulfonates
We claim: 1. A method of inhibiting fungi or bacteria pathogenic to plants which comprises applying to said fungi, bacteria or the locus thereof a biocidally effective amount within the range of about... Read More
Inventors: Smith, deceased, Herbert Q.; Smith, legal representative, by Jacqueline; Toukan, Sameeh Said;, Assignee: Pennwalt Corporation (Philadelphia, PA) |
New O-(3-amino-2-hydroxy-propyl)-amidoxime derivatives, process for the preparation thereof and pharmaceutical compositions containing same
What we claim is: 1. A compound of the formula I or a pharmaceutically acceptable acid addition salt thereof ##STR9## wherein R.sup.2 and R.sup.3 are polymethylene which together form a five- to eight... Read More
Inventors: Takacs, Kalman; Literati, Peter N.; Kiss nee Ajzert, Ilona; Simay, Antal; Szentivanyi, Matyas; Virag, Sandor; Farago, Katalin;, Assignee: Chinoin Gyogyszer es Vegyeszeti Termekek Gyara R.T. (Budapest, HU) |
Pharmacologically active compositions
What we claim is: 1. A synergistic pharmaceutical composition for use as an anti-allergic comprising a compound of formula (I) ##STR5## wherein Z is oxygen or carbonyl and Z is carboxyl or 5-tetrazoly... Read More
Inventors: Garland, Lawrence George; Follenfant, Michael John; Tateson, James Edward;, Assignee: Burroughs Wellcome Co. (Raleigh, NC) |
Preparation of N-(aminoalkyl)piperazine
What is claimed is: 1. A process for producing an N-(aminoalkyl)piperazine compound directly from a piperazine compound selected from piperazine and C-(substituted) piperazine wherein the substituents... Read More
Inventors: Brennan, Michael E.; Moss, Philip H.; Yeakey, Ernest L.;, Assignee: Texaco Development Corporation (New York, NY) |
4-(4'-Hydroxycyclohexyl)-2,2,6,6-tetramethyl piperidines
We claim: 1. A compound having the formula: ##SPC12## wherein R.sub.1, R.sub.2, R.sub.3 and R.sub.4 are the same or different and each is hydrogen, an alkyl having from 1 to 9 carbon atoms, a cycloalk... Read More
Inventors: Smith, Malcolm John; Randell, Donald Richard;, Assignee: Ciba-Geigy Corporation (Ardsley, NY) |
Preparation of alkanedisulfonates from olefins using carboxylic acid
Suitable olefins for use in my process contain from 2 to about 40 carbon atoms, preferably from about 10 to about 36 carbon atoms. Preferably, the olefins are linear. Also, the double bond can be eit... Read More
Inventors: Convers, Ronald J.;, Assignee: Continental Oil Company (Ponca City, OK) |
Substituted thio-substituted benzyl-propionyl-L-prolines
OF THE INVENTION The novel substituted .omega.-aroyl(propionyl or butyryl)-L-prolines and esters thereof of the present invention are generally obtainable as white to yellow crystalline materials hav... Read More
Inventors: McEvoy, Francis J.; Albright, Jay D.;, Assignee: American Cyanamid Company (Stamford, CT) |
Method for industrial production of N-substituted dipropylacetamides
We claim: 1. A compound having the formula ##EQU3## wherein R is 2-picolyl, 3-picolyl or 4-picolyl. 2. A compound as claimed in claim 1, in which R is 2-picolyl. 3. A compound as claimed in claim 1, i... Read More
Inventors: Martinez Roldan, Christobal; Fernandez Brana, Miguel; Castellano Berlanga, Jose Maria;, Assignee: Laboratorios Made, S.A. (Madrid, ES) |
Analgesic compositions containing 1,2-dihydro-2-oxoquinol-4-ylpropionic acid derivatives
What we claim is: 1. A pharmaceutical analgesic composition which comprises a quinolone alkanoic acid of the formula ##STR53## wherein A is a methylene, ethylene or propenylene; R.sup.1 is hydrogen; R... Read More
Inventors: Brittain, David R.; Brown, Edward D.; Hepworth, Walter; Stacey, Gilbert J.;, Assignee: Imperial Chemical Industries Limited (London, GB2) |
2-Naphthyl-lower-alkanoylamines
INCLUSIVE OF THE PREFERRED EMBODIMENTS More specifically, the invention relates to a 2-naphthyl-lower-alkylamines, which are useful as anti-inflammatory agents, having the formula: ##STR1## where R.s... Read More
Inventors: Zenitz, Bernard L.;, Assignee: Sterling Drug Inc. (New York, NY) |
Metal salts of 1,1,5,5-tetrasubstituted dithiobiurets as population control agents
What I claim and desire to protect by Letters Patent is: 1. A method of inhibiting ovulation in a female mammal, which comprises orally administering to that mammal at least for a period of time prior... Read More
Inventors: Diveley, William R.;, Assignee: Hercules Incorporated (Wilmington, DE) |
Piperidine derivatives
I claim: 1. A compound of the formula ##SPC18## wherein n is 1, 2, 3 or 4, Y is hydrogen or a straight- or branched alkyl residue having from 1 to 12 carbon atoms, an alkenyl residue having from 3 to ... Read More
Inventors: Cook, Barry;, Assignee: Ciba-Geigy Corporation (Ardsley, NY) |
4-Hydroxy-3-nitro-carbostyril compounds
We claim: 1. A compound of the formula (IA) or a pharmaceutically acceptable salt thereof: ##STR6## wherein one of the groups R.sub.6, R.sub.7 and R.sub.8 are hydrogen and the other two are methyl, et... Read More
Inventors: Buckle, Derek Richard; Cantello, Barrie Christian Charles; Smith, Harry;, Assignee: Beecham Group Limited (GB) |
Vitamin E orotate and a method of producing the same
What we claim is: 1. Vitamin E orotate consisting of a tocopheryl moiety selected from .alpha.-, .beta.-, .gamma.- and .delta.-tocopheryl groups and an unsubstituted orotyl moiety combined with said t... Read More
Inventors: Hasunuma, Kyotaro; Kurokawa, Masahiro; Abe, Takashi;, Assignee: Kanebo Ltd. (Tokyo, JA) |
Treatment of liver dysfunction with 2-amino-6-benzyl-3-ethoxycarbonyl-4,5,6,7-tetrahydro-thieno[2,3-c]pyridi ne hydrochloride
OF THE INVENTION The present invention has been accomplished on the basis of new finding that tinoridine hydrochloride shows highly protective effects on liver injuries of animals caused by carbon te... Read More
Inventors: Kobayakawa, Toshihiro; Yasuda, Hiroshi; Goto, Kazuhiro; Nakanishi, Michio;, Assignee: Yoshitomi Pharmaceutical Industries, Ltd. (Osaka, JA) |
Intravitreal medicine delivery
Intravitreal Medicine Delivery Device- First Embodiment The first embodiment of an intravitreal medicine delivery device of the resent invention is identified in FIGS. 1-6 by the numeral 30 and is sh... Read More
Inventors: Avery, Robert Logan; Luttrull, Jeffrey Kevin;, Assignee: |
Deodorant and antimicrobial dispersions
OF THE INVENTION AND PREFERRED EMBODIMENTS The present invention will next be described more specifically based on preferred embodiments. The deodorant and antimicrobial component, which makes up the... Read More
Inventors: Hoshino, Akira; Saji, Mikio; Hayashi, Kozaburo;, Assignee: Dainichiseika Color & Chemicals Mfg. Co, Ltd. (Tokyo, JP) |
Process for hypotensive 4-amino-2-(piperazin-1-yl) quinazoline derivatives
OF THE INVENTION As indicated before, the object of the instant invention is to provide a process for the preparation of compounds of formula I, by reaction of a compound of formula II, or a salt the... Read More
Inventors: Hess, Hans-Jurgen E.;, Assignee: Pfizer Inc. (New York, NY) |
Child-resistant safety belt buckle
Referring to FIG. 1, a push-button safety belt buckle 1 is shown comprising a metal body 2 that is connected to one end 3 of a segment safety belt 4 or harness and a leaf or tongue 5 that is connecte... Read More
Inventors: Hunter, Robert M.; Hunter, Mary M.;, Assignee: |
Synthetic compounds and compositions with enhanced cell binding
In one aspect of the present invention, a family of synthetic peptides are provided that mimic the cell binding domain of collagen so that these compounds competitively inhibit the binding of cells to... Read More
Inventors: Bhatnagar, Rajendra S.;, Assignee: The Regents of the University of California (Oakland, CA) |
Substituted fusaric acid derivatives
OF THE PREFERRED EMBODIMENTS The halo-fusaric acid amides of this invention have the formula: ##SPC3## Wherein X represents hydrogen or halogen atom; and Y represents a halogen atom; R.sub.1 and R.su... Read More
Inventors: Miyano, Tetsuji; Suzuki, Kunio; Fukatsu, Hiroshi;, Assignee: Banyu Pharmaceutical Co., Ltd. (Nagoya, JA) |
Preparation of 5,8-methano-5H-benzocyclohepten-10-amines
The subject matter which the applicant regard as their invention is particularly pointed out and distinctly claimed as follows: 1. A process for the preparation of a chemical compound of the formula: ... Read More
Inventors: Freed, Meier E.; Potoski, John R.;, Assignee: American Home Products Corporation (New York, NY) |
Preparation of piperidinyl-alkyl-benzamides
I claim: 1. Piperidinyl-alkyl-benzamides having the general formula ##STR5## wherein R is hydrogen, an alkyl group having from 1 to 4 carbon atoms, an alkoxy group having from 1 to 4 carbon atoms, hal... Read More
Inventors: Roll, William D.;, Assignee: The University of Toledo (Toledo, OH) |
Naphthylethylureas and naphthylethylthioureas
We claim: 1. A compound selected from those of formula I: ##STR4## in which: R represents hydrogen or a group OR.sub.3 wherein R.sub.3 represents straight-chained or branched alkyl having 1 to 6 carbo... Read More
Inventors: Lesieur, Daniel; Yous, Said; Depreux, Patrick; Adam, Gerard; Renard, Pierre; Pfeiffer, Bruno; Guardiola-Lemaitre, Beatrice;, Assignee: Adir et Compagnie (Courbevoie, FR) |
Naphthylethylureas and naphthylethylthioureas
We claim: 1. A method of treating a mammal afflicted with a disorder of the melatoninergic system selected from sleep and seasonal disorders comprising the step of administering to the said mammal an ... Read More
Inventors: Lesieur, Daniel; Yous, Said; DePreux, Patrick; Adam, Gerard; Renard, Pierre; Pfeiffer, Bruno; Guardiola-Lemaitre, Beatrice;, Assignee: Adir et Compagnie (Courbevoie, FR) |
Trisubstituted naphthylalkylamides for disorders of the melatoninergic system
We claim: 1. A compound of formula (I): ##STR28## in which: R represents hydrogen or a radical chosen from alkyl, substituted alkyl and --O--R'; with R' representing hydrogen or a radical selected fro... Read More
Inventors: Depreux, Patrick; Mansour, Hamid A.; Lesieur, Daniel; Lefoulon, Fran.cedilla.ois; Renard, Pierre; Adam, Gerard; Delagrange, Philippe;, Assignee: Adir et Compagnie (Courbevoie, FR) |
Potent inducers of terminal differentiation and method of use thereof
OF THE INVENTION The invention provides a class of compounds having the structure: [R--A]--B--A.sub.1 --B.sub.1 --[A.sub.2 --B.sub.2 --].sub.a [A.sub.3 --B.sub.3 --].sub.b [A.sub.4 --R.sub.1 ] wherei... Read More
Inventors: Breslow, Ronald; Marks, Paul A.; Rifkind, Richard A.;, Assignee: The Trustees of Columbia University in the City of New York (New York, NY); Sloan-Kettering Institute for Cancer Research (New York, NY) |
Production of propionic acid
What is claimed is: 1. A one-step process for the preparation of propionic acid which comprises reacting ethylene with carbon monoxide and water at a temperature of 50.degree. C to 300.degree. C and a... Read More
Inventors: Paulik, Frank E.; Hershman, Arnold; Roth, James F.; Craddock, John H.;, Assignee: Monsanto Company (St. Louis, MO) |
1-Ethyl-1-(alkoxycarbonylethyl)-octahydro-indolo[2,3-a]quinolizines
What we claim is: 1. 1.alpha.-Ethyl-1-(sec-butoxycarbonyl-ethyl)-1,2,3,4,6,7,12, 12b.alpha.-octahydro-indolo[2,3-a]quinolizine. 2. 1.alpha.-Ethyl-1-(sec-butoxycarbonyl-ethyl)-1,2,3,4,6,7,12, 12b.beta.... Read More
Inventors: Szantay, Csaba; Szabo, Lajos; Kalaus, Gyorgy; Karpati, Egon; Szporny, Laszlo;, Assignee: Richter Gedeon Vegyeszeti Gyar Rt. (Budapest, HU) |
Saccharase inhibiting 3,4,5-trihydroxypiperidine derivatives
What is claimed is: 1. A 3,4,5-trihydroxypiperidine derivative of the formula ##STR99## or a pharmaceutically acceptable salt thereof, in which R.sub.1 denotes a hydrogen atom, an amino group, an alky... Read More
Inventors: Stoltefuss, Jurgen; Muller, Lutz; Puls, Walter; Sitt, Rudiger;, Assignee: Bayer Aktiengesellschaft (Leverkusen, DE) |
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Vasodialators 
